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BS168256
BIO-X

SET2 NEW

Inhibitor of the transient receptor vanilloid channel, specific for the TRPV2 subtype with IC50 value of 0.46 μM. In human prostate cancer cells, SET2 inhibited cell migration but did not affect cell survival. SET2 has been proposed as a potential anti-cancer and anti-metastatic agent.

Technical Data

Synonyms: N-(Furan-2-ylmethyl)-3-((4-(N'-methyl-N'-propylamino)-6-(trifluoromethyl)-pyrimidin-2-yl)thio)-propanamide.
Product Code: BS168256
Chemical Formula: C17H21F3N4O2S
Molecular Weight: 402.44

References


  • Chai et al (2019). Structure-Based Discovery of a Subtype-Selective Inhibitor Targeting a Transient Receptor Potential Vanilloid Channel. Journal of Medicinal Chemistry 62(3):1373-1384.

Solubility

Stability

Further Information


Datasheets

Specification: View
MSDS: View

Synonyms:
N-(Furan-2-ylmethyl)-3-((4-(N'-methyl-N'-propylamino)-6-(trifluoromethyl)-pyrimidin-2-yl)thio)-propanamide.
Chemical Formula:
Molecular Weight:
402.44
Product Structure
References:
1. Chai et al (2019). Structure-Based Discovery of a Subtype-Selective Inhibitor Targeting a Transient Receptor Potential Vanilloid Channel. Journal of Medicinal Chemistry 62(3):1373-1384.
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