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BA167283
BIO-X

AP 202

Selective antagonist of α4β2 nicotinic acetylcholine receptors (nAChRs), selective over α4β4, α3β2, and α3β4α5 nAChRs. Lowers nicotine self-administration in vivo for 30 minutes. Inhibits nicotine seeking, following relapse, during both prime- and cue-induced reinstatement. 

Technical Data

CAS No: 2196197-89-2
Product Code: BA167283
Chemical Formula: C11H16N4
Molecular Weight: 204.27

References


  • Wu J et al (2017). Highly Selective and Potent α4β2 nAChR Antagonist Inhibits Nicotine Self-Administration and Reinstatement in Rats. J Med Chem 60(24):10092-10104.

Solubility

Stability

Further Information


Datasheets


AP 202 - Bio-X

CAS No:
2196197-89-2
Chemical Formula:
Molecular Weight:
204.27
Product Structure
References:
1. Wu J et al (2017). Highly Selective and Potent α4β2 nAChR Antagonist Inhibits Nicotine Self-Administration and Reinstatement in Rats. J Med Chem 60(24):10092-10104.

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