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BS166447

SR 16832 - Bio-X

Inhibits binding of endogenous ligands to peroxisome proliferator-activated receptor gamma (PPARγ), blocking its activation and transcription. Unlike orthosteric antagonists GW 9662 and T 0070907, SR 16832 blocks both allosteric and orthosteric activation of PPARγ.

Technical Data

CAS No: 2088135-12-8
Product Code: BS166447
Chemical Formula: C17H12ClN3O4
Molecular Weight: 357.75

References


  • Brust R et al (2017). Modification of the Orthosteric PPARγ Covalent Antagonist Scaffold Yields an Improved Dual-Site Allosteric Inhibitor. ACS Chem Biol 12(4):969-978.

Solubility

Stability

Further Information


Datasheets


SR 16832 - Bio-X

CAS No:
2088135-12-8
Chemical Formula:
Molecular Weight:
357.75
Product Structure
References:
1. Brust R et al (2017). Modification of the Orthosteric PPARγ Covalent Antagonist Scaffold Yields an Improved Dual-Site Allosteric Inhibitor. ACS Chem Biol 12(4):969-978.

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