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7-TM Receptors

A large proportion of commercially-available drugs target seven transmembrane (7-TM) receptors, of which a selection is offered by Carbosynth that are listed below.  7-TM receptors are the largest superfamily of cell surface receptors, also known as G-protein-coupled receptors (GPCRs). These receptors transduce signals from the extracellular space to the cytoplasm, via their transmembrane domains. Based on sequence homology, 7-TM receptors are classed into 6 groups: Class A (rhodopsin-like), Class B (secretin receptor family), Class C (metabotropic glutamate), Class D (fungal mating pheromone receptors), Class E (cyclic AMP receptors) and Class F (frizzled/smoothened).

Code Cas No Product Description
BF166977 1364933-62-9

5F-AB 001

Synthetic cannabinoid analog
BM166976 895155-25-6

AB 005

Synthetic cannabinoid
FM61417 22972-55-0


GPR55 agonist
FA16904 447407-36-5

AC 42

Muscarinic (M1) receptor agonist
BA17966 220556-69-4


Cannabinoid (CB1) receptor agonist
BA166874 51037-30-0


Niacin receptor 1 (NIACR1) antagonist; lipid lowering
FA31012 320345-99-1

Aclidinium bromide

Muscarinic antagonist; bronchodilator
BA17967 229021-64-1


CB1 cannabinoid receptor agonist
FA103122 851881-60-2

ADX 47273

Positive allosteric modulator of mGlu5 receptors
BA166488 851881-59-9

(R)-ADX 47273

Inhibits metabotropic glutamate receptor (mGluR5)
BA167079 138112-76-2


Melatonin agonist; 5-HT2B and 5-HT2C serotonin receptor antagonist
BA164142 79561-22-1

Alarelin Acetate

Gonadotropin-releasing hormone agonist
BA164143 18559-94-9


β2-adrenergic receptor agonist; bronchodilator
FA17263 50293-90-8

(R)-Albuterol hydrochloride

β2-adrenergic receptor agonist; bronchodilator
BA164388 51022-70-9

Albuterol sulfate

β-adrenergic receptor agonists
BA164145 81403-80-7


α-adrenoceptor antagonist; treatment for benign prostatic hyperplasia
FA150825 59338-87-3

Alizapride hydrochloride

Dopamine (D2) receptor antagonist
BA166116 913358-93-7

Almorexant hydrochloride

Antagonist of orexin receptors OX1 and OX2
FA17315 154323-46-3

Almotriptan hydrochloride

Serotonin (5-HT) receptor agonist
BA166465 122852-69-1

Alosetron hydrochloride

Serotonin 5-HT3 receptor antagonist
FA31828 745-65-3


Inhibits platelet aggregation; vasodilator
BA164152 156053-89-3


Peripheral μ-opioid receptor antagonist; gastroprokinetic
BA17338 183232-66-8

AM 251 NEW

CB1 cannabinoid receptor antagonist
BA164153 177036-94-1


Endothelin A receptor antagonist; anti-hypertensive
FA148913 155148-31-5

AMD 3100 octahydrochloride

Chemokine receptor CXCR4 antagonist
BA164158 71675-85-9


Dopamine D2/D3 receptor antagonist; anti-psychotic;
BA164170 14028-44-5


Serotonin (5-HT2) receptor antagonist; inhibits norepinephrine reuptake
FA138836 2706-50-5

DL-Amphetamine hydrochloride

Analytic reference standard
FA162453 51-63-8

(+)-Amphetamine sulphate

Inhibits reuptake of catecholamines; stimulates central nervous system
BA166586 94421-68-8


Endogenous cannabinoid and TRPV1 receptor agonist
FA17951 105219-56-5


Platelet-activating factor antagonist
BA165146 1268881-20-4

APD 371

Cannabinoid receptor CB2 agonist
BA166505 461443-59-4


Inhibits chemokine receptor CCR5; anti-viral activity against HIV
BA164186 73218-79-8

Apraclonidine hydrochloride

α2-adrenoceptor agonist; anti-glaucoma agent
BA164216 170729-80-3


Antagonist of neurokinin-1 receptor; anti-emetic
BA165448 733750-99-7

AR 231453

A potent and selective small molecule agonist of GPR119
BA164218 129722-12-9


Partial agonist of dopamine (D2) and serotonin (5-HT1A) receptors
BA45604 128007-31-8


CB1 cannabinoid receptor and vanilloid TRPV1 (VR1) agonist
FA17998 65576-45-6


Inhibits dopamine, serotonin and adrenergic receptors
FA61540 85650-56-2

Asenapine maleate

Inhibits dopamine, serotonin and adrenergic receptors
FA18002 68844-77-9


Histamine-1 receptor antagonist; hERG K+ channel blocker
BA166036 29122-68-7


β-adrenoceptor blocker
FA64946 104075-48-1

Atipamezole HCl

α2-adrenoceptor antagonist
FA40914 914453-95-5

Atosiban acetate

Oxytocin receptor antagonist
FA29947 173937-91-2


Endothelin receptor antagonist
FA64949 195733-43-8

Atrasentan hydrochloride

Endothelin receptor antagonist
BA164232 79307-93-0

Azelastine hydrochloride

Histamine-1 receptor antagonist; NFκB activator
BA164233 147403-03-0


Angiotensin II, type I receptor antagonist; anti-hypertensive
FB18126 66514-99-6


GABA(B) agonist; anti-spastic agent; skeletal muscle relaxant
BB166152 1134-47-0


GABA(B) agonist; anti-spastic agent; skeletal muscle relaxant
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