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Ion Channels

Ion channels are transmembrane proteins with the ability to control ion currents across cell membrane. They are essential for maintaining resting membrane potential as well as for generation of action potentials in neurons, muscle and endocrine cells. Our collection of ion channel modulators include blockers of ligand-gated and voltage-gated channels, as well as mechanosensitive, cyclic nucleotide-gated channels and more.

Code Cas No Product Description
BE166951 945828-50-2

AA 29504

Allosteric GABAA receptor modulator; anxiolytic
BA164134 77337-73-6

Acamprosate calcium

GABA receptor agonist; threatment for alcohol dependence
BA165790 865305-30-2

AF 353

Antagonist of P2X3/P2X2/3 purinoreceptors
BA166015

Ambroxol HCl

Antioxidant; secretolytic; anti-inflammatory; sodium channel blocker
FA164880 545395-94-6

AMG 9810

Vanilloid receptor 1 antagonist
FA61531 17440-83-4

Amiloride HCl

Sodium channel inhibitor; inhibitor of urokinase-type plasminogen activator
BA139263 1951-25-3

Amiodarone HCl

Multi-channel blocker; anti-arrhythmic agent
BA164164 88150-42-9

Amlodipine base

Inhibits L-type calcium channels; anti-hypertensive; antianginal
BA164162 111470-99-6

Amlodipine besylate

Inhibits L-type calcium channels; anti-hypertensive; antianginal
BA164165 88150-47-4

Amlodipine maleate

Inhibits L-type calcium channels; anti-hypertensive; antianginal
BA165665 926023-82-7

AMTB NEW

TRPM8 channel blocker
FA17896 3471-05-4

Anabaseine

Natural neurotoxin
BA164183 72432-10-1

Aniracetam

AMPA/kainate desensitization inhibitor
FA145501 178419-42-6

AR-R 17779 hydrochloride

Agonist of α7 nicotinic receptor
FA52437 14923-17-2

Arcaine Sulfate

Antagonist of NMDA receptor
FA18027 64228-81-5

Atracurium besylate

Nicotinic AChR antagonist; neuromuscular blocking agent; muscle relaxant
FA18062 123040-69-7

Azasetron hydrochloride

Serotonin 5-HT3 receptor antagonist; anti-emetic
FA158515 345303-91-5

AZD 9056 HCl

P2X7 receptor antagonist
FB18144 104757-53-1

Barnidipine hydrochloride

Calcium channel blocker
BB162780 71145-03-4

BAY K 8644

Activates L-type Ca2+ channels; vasoconstrictive
BB165272 393514-24-4

BCTC

Antagonist of vanilloid receptor TRPV1 
FB64953 91599-74-5
105979-17-7

Benidipine hydrochloride

Calcium channel blocker 
BB164251 485-49-4

(+)-Bicuculline

Inhibitor of ionotropic receptor GABA(A)
BB162664 40709-69-1

(-)-Bicuculline methiodide

Inhibitor of ionotropic receptor GABA(A); less active isomer
FB157252 11032-79-4

alpha-Bungarotoxin

Antagonist of nicotinic acetylcholine receptors; neurotoxin
BB166160 2180-92-9

Bupivacaine

Sodium channel blocker, targets channel intracellular domain
BC166161 298-46-4

Carbamazepine

GABA agonist; voltage-gated sodium channel blocker
FC19680 36507-30-9

Carbamazepine 10,11-epoxide

Inhibitor of neuronal voltage-gated sodium channels
FC158497 724424-43-5

CE 224,535

Antagonist of purinoreceptor P2X7
BC164300 58-25-3

Chlordiazepoxide

Benzodiazepine derivative; hypnotic; anxiolytic; anti-convulsant; sedative
BC164309 132203-70-4

Cilnidipine

Inhibits L- and N-type calcium channels; anti-hypertensive; neuroprotective
BC167081 298-57-7

Cinnarizine

Calcium channel blocker; piperazine derivative
FC74963 92953-10-1

Clofilium tosylate

Potassium channel blocker; anti-arrhythmic; cardiac depressant
FC20628 115066-14-3

CNQX

Glutamate antagonist
FC109903 106375-28-4

Omega-Conotoxin GVIA trifluoroacetate salt

Inhibitor of N-type voltage-gated calcium channels
FC20595 215923-54-9

CX 546

AMPA receptor potentiator
BC164343 485-35-8

Cytisine

Nicotinic ACh receptor agonist
BD162474 79055-68-8

D-AP5

Antagonist of NMDA receptor
BD162627 29734-68-7

Dihydro-b-erythroidine HBr

Antagonist of nicotinic receptor
BD166408 33286-22-5

Diltiazem

L-type calcium channel blocker
BD162539 76326-31-3

DL-AP5

Antagonist of NMDA receptor
FD22437 2379-57-9

DNQX

AMPA/ kainate receptor antagonist 
BD164377 115256-11-6

Dofetilide

Potassium channel blocker; antiarrhythmic agent
FD14809 115956-13-3

Dolasetron mesylate

Serotonin receptor 5-HT3 antagonist
FD61522 113-07-5

Doxapram hydrochloride

Inhibitor of TASK tandem pore potassium channel; respiratory stimulant
BD164395 141625-93-6

Dronedarone hydrochloride

Multichannel blocker; reduces sodium and calcium currents
FE22688 105816-05-5

ent-nateglinide

Blocker of ATP-dependent potassium channels; insulinotropic agent
FE156792 138729-47-2

Eszopiclone

Modulator of GABA(A) receptors
FE162097 1262780-97-1

Etelcalcetide

Agonist of calcium sensing receptor CASR; calcimimetic agent
FF23236 119945-59-4

(R)-(+)-Felodipine

Voltage-gated calcium channel blocker
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