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Ion Channels

Ion channels are transmembrane proteins with the ability to control ion currents across cell membrane. They are essential for maintaining resting membrane potential as well as for generation of action potentials in neurons, muscle and endocrine cells. Our collection of ion channel modulators include blockers of ligand-gated and voltage-gated channels, as well as mechanosensitive, cyclic nucleotide-gated channels and more.

Code Cas No Product Description
BE166951 945828-50-2

AA 29504

Allosteric GABAA receptor modulator; anxiolytic BIO-X
BA164134 77337-73-6

Acamprosate calcium

GABA receptor agonist; threatment for alcohol dependence BIO-X
BA165790 865305-30-2

AF 353

Antagonist of P2X3/P2X2/3 purinoreceptors BIO-X
BA166177 665-66-7

Amantadine hydrochloride

NMDA receptor antagonist; anti-viral; anti-Parkinsonian BIO-R
BA166015 23828-92-4

Ambroxol hydrochloride

Antioxidant; secretolytic; anti-inflammatory; sodium channel blocker BIO-R
FA164880 545395-94-6

AMG 9810

Vanilloid receptor 1 antagonist BIO-X
FA61531 17440-83-4

Amiloride hydrochloride

Sodium channel inhibitor; inhibitor of urokinase-type plasminogen activator BIO-R
BA139263 19774-82-4

Amiodarone hydrochloride

Multi-channel blocker; anti-arrhythmic agent BIO-R
BA164164 88150-42-9

Amlodipine

Inhibits L-type calcium channels; anti-hypertensive; antianginal BIO-R
BA164162 111470-99-6

Amlodipine besylate

Inhibits L-type calcium channels; anti-hypertensive; antianginal BIO-X
BA164165 88150-47-4

Amlodipine maleate

Inhibits L-type calcium channels; anti-hypertensive; antianginal BIO-R
BA165665 926023-82-7

AMTB NEW

TRPM8 channel blocker BIO-X
FA17896 3471-05-4

Anabaseine

Natural neurotoxin BIO-X
BA164183 72432-10-1

Aniracetam

AMPA/kainate desensitization inhibitor BIO-R
BA167283 2196197-89-2

AP 202

α4β2 nAChR antagonist; reduces nicotine self-administration in vivo BIO-X
FA145501 178419-42-6

AR-R 17779 hydrochloride

Agonist of α7 nicotinic receptor BIO-X
FA18062 123040-69-7

Azasetron hydrochloride

Serotonin 5-HT3 receptor antagonist; anti-emetic BIO-X
FA158515 345303-91-5

AZD 9056 hydrochloride

P2X7 receptor antagonist BIO-X
FB18144 104757-53-1

Barnidipine hydrochloride

Calcium channel blocker BIO-X
BB162780 71145-03-4

BAY K 8644

Activates L-type Ca2+ channels; vasoconstrictive BIO-X
BB165272 393514-24-4

BCTC

Antagonist of vanilloid receptor TRPV1  BIO-X
FB64953 91599-74-5

Benidipine hydrochloride

Calcium channel blocker  BIO-X
BB164251 485-49-4

(+)-Bicuculline

Inhibitor of ionotropic receptor GABA(A) BIO-X
BB162664 40709-69-1

(-)-Bicuculline methiodide

Inhibitor of ionotropic receptor GABA(A); less active isomer BIO-X
FB157252 11032-79-4

alpha-Bungarotoxin

Antagonist of nicotinic acetylcholine receptors; neurotoxin BIO-X
BB166160 2180-92-9

Bupivacaine

Sodium channel blocker, targets channel intracellular domain BIO-R
BC166161 298-46-4

Carbamazepine

GABA agonist; voltage-gated sodium channel blocker BIO-R
FC158497 724424-43-5

CE 224535

Antagonist of purinoreceptor P2X7 BIO-X
BC164300 58-25-3

Chlordiazepoxide

Benzodiazepine derivative; hypnotic; anxiolytic; anti-convulsant; sedative BIO-X
BC164309 132203-70-4

Cilnidipine

Inhibits L- and N-type calcium channels; anti-hypertensive; neuroprotective BIO-X
BC167081 298-57-7

Cinnarizine

Calcium channel blocker; piperazine derivative BIO-R
FC74963 92953-10-1

Clofilium tosylate

Potassium channel blocker; anti-arrhythmic; cardiac depressant BIO-X
FC20628 115066-14-3

CNQX

Glutamate antagonist BIO-X
FC109903 106375-28-4

Omega-Conotoxin GVIA trifluoroacetate salt

Inhibitor of N-type voltage-gated calcium channels
BC168104 126453-07-4

(R)-CPP

NMDA receptor antagonist
FC20595 215923-54-9

CX 546

AMPA receptor potentiator BIO-X
BC164343 485-35-8

Cytisine

Partial agonist of nAChRs; aids smoking cessation BIO-X
BD162474 79055-68-8

D-AP5

Antagonist of NMDA receptor BIO-X
BD162627 29734-68-7

Dihydro-b-erythroidine hydrobromide

Antagonist of nicotinic receptor BIO-X
BD166408 33286-22-5

Diltiazem

L-type calcium channel blocker BIO-R
BD162539 76326-31-3

DL-AP5

Antagonist of NMDA receptor BIO-X
FD22437 2379-57-9

DNQX

AMPA/ kainate receptor antagonist  BIO-X
BD164377 115256-11-6

Dofetilide

Potassium channel blocker; antiarrhythmic agent BIO-X
FD14809 115956-13-3

Dolasetron mesylate

Serotonin receptor 5-HT3 antagonist BIO-X
FD61522 113-07-5

Doxapram hydrochloride

Inhibitor of TASK tandem pore potassium channel; respiratory stimulant BIO-X
BD164395 141625-93-6

Dronedarone hydrochloride

Multichannel blocker; reduces sodium and calcium currents BIO-X
FE156792 138729-47-2

Eszopiclone

Modulator of GABA(A) receptors
FF23236 119945-59-4

(R)-(+)-Felodipine

Voltage-gated calcium channel blocker
BF164445 72509-76-3

Felodipine

L-type calcium channel blocker; anti-hypertensive BIO-X
BF160700 78538-74-6

FG 7142

Agonist of benzodiazepine receptor; anxiogenic BIO-X
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